Svaki ml Testo Rapid sadrži dovoljno Testosteron Propionate 100mg u uljnoj bazičnoj količini. Testosteron se izlučuje iz Leydigove ćelije testisa. Odgovorna je za razvoj sekundarnih spolnih znakova kod muškaraca u vrijeme puberteta i naknadno održavanje spermatogeneze tokom reproduktivnog života muškaraca. Veže se za intraćelijske receptore u ciljanim ćelijama gde kompleks hormonskih receptora prelazi u jezgro gde se vezuje za specifična mesta vezivanja na hromozomima. To dovodi do povećane sinteze mRNA i proteina.

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